Corrigendum: Progress in antiandrogen design targeting hormone binding pocket to circumvent mutation based resistance
نویسندگان
چکیده
[This corrects the article on p. 57 in vol. 6, PMID: 25852559.].
منابع مشابه
Progress in antiandrogen design targeting hormone binding pocket to circumvent mutation based resistance
Androgen receptor (AR) plays a critical role in the development and progression of prostate cancer (PCa). Current clinically used antiandrogens such as flutamide, bicalutamide, and newly approved enzalutamide mainly target the hormone binding pocket (HBP) of AR. However, over time, drug resistance invariably develops and switches these antiandrogens from antagonist to agonist of the AR. Accumul...
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عنوان ژورنال:
دوره 6 شماره
صفحات -
تاریخ انتشار 2015